首页 工具
登录
购物车

搜索结果

Search Results for " nk receptor "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T23316 SB 218795

Neurokinin receptor GPCR/G Protein; Neuroscience
SB 218795 是一种有效的特异性 NK3 拮抗剂,对 hNK3 的 Ki 为 13 nM,比 hNK2 和 hNK1 的特异性高约 90 倍和 7000 倍。
T7633 Senktide

Neurokinin receptor GPCR/G Protein; Neuroscience
Senktide 是速激肽NK3受体激动剂。
T16849 SB-222200

Neurokinin receptor GPCR/G Protein; Neuroscience
SB-222200 是一种选择性口服活性的,具有血脑屏障渗透性的 NK-3 受体拮抗剂,用于中枢神经系统疾病的研究。
TP1087 Substance P

Neurokinin P,P物质

Endogenous Metabolite; Neurokinin receptor GPCR/G Protein; Metabolism; Neuroscience
Substance P (Neurokinin P) 是一种神经肽,其内源性受体是神经激肽1受体,在中枢神经系统中作为神经递质和神经调节剂。
TP1572 GR-73632

Neurokinin receptor GPCR/G Protein; Neuroscience
GR-73632 强效和选择性速激肽 NK1 受体激动剂,可通过传递瘙痒信号的 NK1 受体直接作用于初级感觉神经元的外周末端。
T7209 Maropitant

马罗匹坦,马罗皮坦

Neurokinin receptor GPCR/G Protein; Neuroscience
Maropitant 是一种可口服的选择性神经激肽受体拮抗剂,通过阻止催吐中心与化学感受器触发区中 P 物质的结合而起作用,有预防呕吐作用。
T38144 Elinzanetant

Neurokinin receptor GPCR/G Protein; Neuroscience
Elizanetant 是有效的神经激肽受体拮抗剂,在精神分裂症研究中有价值。
T15278 Fezolinetant

ESN-364

Neurokinin receptor GPCR/G Protein; Neuroscience
Fezolinetant (ESN-364) 是一种神经激肽-3 受体拮抗剂,可用于更年期潮热的研究。
T7549 Talnetant

SB 223412

Neurokinin receptor GPCR/G Protein; Neuroscience
Talnetant (SB 223412) 是一种选择性、竞争性、脑渗透性 NK3 受体拮抗剂,Ki 为1.4 nM。它比对hNK-2受体的抑制性高100倍,具有调节中脑边缘和中脑皮质多巴胺能神经传递的能力。
TP1883 [Lys5,MeLeu9,Nle10]-NKA(4-10)

Neurokinin receptor GPCR/G Protein; Neuroscience
[Lys5,MeLeu9,Nle10]-NKA(4-10) 是高选择性和强效 NK2 受体激动剂,IC50值为 6.1 nM,可诱导大鼠眼底和膀胱收缩,EC50 值分别为 117 和 10 nM。
T8235 L-732138

Neurokinin receptor GPCR/G Protein; Neuroscience
L-732138 是选择性有效和竞争性神经激肽-1受体拮抗剂,IC50为 2.3 nM,可减轻痛觉过敏并具有抗肿瘤作用。它在克隆的人 NK-1受体中的效力比在克隆大鼠 NK-1受体中高 200 倍,比人类 NK-2 和 NK-3 受体高 1000 倍以上。
T17156 Tradipitant

VLY-686,LY686017

Neurokinin receptor GPCR/G Protein; Neuroscience
Tradipitant (VLY-686) 是一种有效的神经激肽-1 拮抗剂。
T7554 Substance P (7-11)

Substance P 7-11(TFA)

Others; Neurokinin receptor GPCR/G Protein; Neuroscience; Others
Substance P (7-11) (Substance P 7-11(TFA)) 是神经肽物质P 的C-末端片段,可引起细胞内钙浓度的增加。
TP1008 Neurokinin A

α-Neurokinin,Substance K,神经激肽A,Neuromedin L

Neurokinin receptor GPCR/G Protein; Neuroscience
Neurokinin A (NKA) 是速激肽家族的一种肽类神经递质,是人体气管道和胃肠道组织中的主要介体,可通过 NK-2受体发挥作用。
T3716 Rolapitant

罗拉吡坦,SCH619734,罗拉匹坦

Neurokinin receptor GPCR/G Protein; Neuroscience
Rolapitant (SCH619734) 是一种高效选择性具有口服活性的神经激肽 1 受体抑制剂,Ki 值为0.66 nM。
T6905 Netupitant

Ro 67-31898/000,奈妥吡坦,CID 6451149

Neurokinin receptor GPCR/G Protein; Neuroscience
Netupitant (CID 6451149) 是一种高效选择性、可口服的神经激肽 1 受体 (NK1) 拮抗剂,具有止吐作用,在 CHO 细胞中对 hNK1的 Ki 值为 0.95 nM。
T13306L Vapreotide acetate

RC-160 acetate,醋酸伐普肽,BMY-41606 acetate

Neurokinin receptor GPCR/G Protein; Neuroscience
Vapreotide acetate (BMY-41606 acetate) 是神经激肽-1 (NK1) 受体拮抗剂,IC50值为 330 nM。
T3034 Eprazinone dihydrochloride

Resplen,Mucitux,Eftapan,NSC 317935,盐酸依普拉酮,依普拉酮二盐酸,Eprazinone 2HCl

Others; Neurokinin receptor GPCR/G Protein; Neuroscience; Others
Eprazinone dihydrochloride (NSC 317935) 是一种具有镇咳和粘液溶解作用的粘液溶解剂。它是神经激肽 1 受体的配体,可改善肺功能和动脉血氧分压,可用于慢性支气管炎的研究。
T1790 Fosaprepitant dimeglumine

福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt

Neurokinin receptor GPCR/G Protein; Neuroscience
Fosaprepitant dimeglumine (MK-0517) 是 Aprepitant 的前药。它是一种神经激肽 1 受体拮抗剂,可用于预防化疗引起的恶心呕吐。
T1743 Aprepitant

MK-869,MK-0869,阿瑞匹坦,L-754030,Aprepitant`

HIV Protease; Antibacterial; Antibiotic; Neurokinin receptor GPCR/G Protein; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Aprepitant (Aprepitant`) 是选择性和高亲和力的神经激肽1受体拮抗剂,Kd 值为86 pM。
T72224 NK1 receptor antagonist 2

NK1receptor antagonist 2 是一种 NK1受体拮抗剂。NK1receptor antagonist 2 可用于耳鸣和听力损失的研究。
T7828 [Sar9,Met(O2)11]-Substance P

Bhsar-sp,NA,精氨酰-脯氨酰-赖氨酰-脯氨酰-谷氨酰-谷氨酰-苯丙氨酰-苯丙氨酰-SAR-亮氨酸-蛋氨酸[O2]-胺

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9,Met(O2)11]-Substance P (NA) 是选择性速激肽NK1受体激动剂。
T7396 Substance P(1-7)

Substance P 1-7

Others; Neurokinin receptor GPCR/G Protein; Neuroscience; Others
Substance P(1-7) (Substance P 1-7) 是神经肽P 物质的片段,可对孤束核产生抑制和缓和作用,具有抗炎、抗伤害和抗痛觉过敏的作用。
T7631 Eledoisin Related Peptide

Eledoisin RP,Eledoisin-Related Peptide,Eledoisin Related Peptide(2TFA)

Neurokinin receptor GPCR/G Protein; Neuroscience
Eledoisin Related Peptide (Eledoisin RP) 是一种速激肽受体配体,是物质P 的类似物,刺激神经元并触发行为反应。
T7559 Neurokinin A(4-10)

神经激肽 A (4-10),Neurokinin A(4-10)(TFA)

Neurokinin receptor GPCR/G Protein; Neuroscience
Neurokinin A(4-10) 是一种速激肽NK2受体激动剂。
T24446L MEN 10207 acetate

Neurokinin receptor GPCR/G Protein; Neuroscience
MEN 10207 acetate 是 NK-2 速激肽受体的选择性拮抗剂。
TP1086 Men 10376 TFA(135306-85-3,free)

Men 10376 TFA,Neurokinin-2 receptor antagonist TFA

Neurokinin receptor GPCR/G Protein; Neuroscience
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) 是一种有效的选择性速激肽 nk-2 受体拮抗剂,对大鼠小肠 nk-2 受体的 K I 值为 4.4 M。
T24697L R 396 acetate

Neurokinin receptor GPCR/G Protein; Neuroscience
R 396 acetate 是一种 NK-2 速激肽受体拮抗剂。
T12000 MEN11467

Neurokinin receptor GPCR/G Protein; Neuroscience
MEN11467 是一种可口服的新型有效且具有选择性的拟肽速激肽 NK 1 受体拮抗剂,可用于研究急性结肠癌。
T69140 Burapitant

SSR 240600

Neurokinin receptor GPCR/G Protein; Neuroscience
Burapitant(SSR 240600)是一种新型非肽速激肽神经激肽 1 (NK) 受体拮抗剂,具有抗焦炉和抗抑郁活性。
T9417L gamma-preprotachykinin amide (72-92) acetate

gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)

Others Others
gamma-preprotachykinin amide (72-92) acetate 是一种 21 个氨基酸的肽,属于速激肽 (TK) 家族,在其 C 末端序列中包括神经激肽 A (NKA)。它对中枢 NK-2 受体的亲和力高于 NKA;它对 NK-1 受体的亲和力较低,但是,它有效地刺激唾液分泌,这是由 NK-1 受体激活介导的。
TP1862L [Sar9] Substance P acetate(77128-75-7 free base)

Neurokinin receptor GPCR/G Protein; Neuroscience
[Sar9] Substance P acetate(77128-75-7 free base) 是一种 NK-1 受体激动剂。 rNK1 特异性激动剂 [Sar-9,Met(O2)11]-SP 模拟了 SP 对孕酮代谢的作用。
T16038 Men 10376

Neurokinin-2 receptor antagonist

CDK Cell Cycle/Checkpoint
Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 μM for rat small intestine NK-2 receptor.
T76405 [D-Trp2,7,9] Substance P

[D-Trp2,7,9] Substance P 是一种速激肽 (Neurokinin Receptor) 拮抗剂,对 NK-1、NK-2和 NK-3受体的 Ki 值分别为 1 μM、1.3 μM 和 ~9 μM。
T70496 MEN-10612

MEN-10612 is a cyclic pseudopeptide and potent tachykinin NK-2 receptor antagonist.
T70243 TAC 363

TAC 363 is a tachykinin NK-2-receptor antagonist.
T12233 NK-1 Antagonist 1

Rolapitant intermediate

Others Others
NK-1 Antagonist 1 is a NK-1 receptor antagonist.
T28706 SCH 206272

SCH206272,SCH-206272

SCH 206272 is a potent, orally active antagonist of tachykinin NK(1), NK(2), and NK(3) receptor.
T75880 GR 94800 TFA

GR 94800 TFA 是有效的、选择性的神经激肽 2(NK2)受体的肽类拮抗剂,其对 NK2、NK1和 NK3受体的 pKB 值分别为 9.6、6.4 和 6.0。
T70497 MEN-10573

MEN-10573 is a cyclic pseudopeptide and potent tachykinin NK-2 receptor antagonist.
T70295 MDL-105212A HCl

MDL-105212A HCl is a nonpeptide NK-1 and NK-2 receptor antagonist.
T29185 YM44781

YM 44781,YM-44781

YM44781 is a non-peptide tachykinin receptor antagonist. YM44781 exhibits high binding affinities at NK(1) (pK(i) = 9.09 +/- 0.02) and NK(2) (pK(i) = 9.94 +/- 0.03) receptors, respectively.
T75879 Men 10376 TFA

Men 10376 TFA 是一种有效的选择性的 tachykinin NK-2受体拮抗剂,对大鼠小肠 NK-2 受体的Ki 值为 4.4 μM。
T29186 YM49598

YM-49598,YM 49598

YM49598 is a tachykinin receptor antagonist. YM49598 exhibited high binding affinities at NK(1) (pK(i) = 9.09 +/- 0.02) and NK(2) (pK(i) = 9.94 +/- 0.03) receptors, respectively. YM49598 was almost inactive but produced a potent inhibition (IC(50) = 11 +/
TQ0087 NKP608

Neurokinin receptor GPCR/G Protein; Neuroscience
NKP608 is a selective and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50: 2.6 nM) and in vivo.
T16406 Orvepitant maleate

GW823296 maleate

Neurokinin receptor GPCR/G Protein; Neuroscience
Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant maleate has the potential for depressive disorder and chronic refractory cough (CRC) treatmen
T70689 MEN-10354

MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.
T76431 GR 83074

GR 83074 是一种有效的选择性 NK-2(Neurokinin Receptor) 拮抗剂,pKB 为 8.23。GR 83074 对 NK-3 没有活性,并表现出 340 倍的 NK-2/NK-1 选择性。
T76454 Substance P (5-11)

Substance P (5-11) 是 Substance P (Substance P ) 的 C 端七肽 ,是一种神经肽,可以与NK-1速激肽受体结合。
T69420 Vestipitant

Vestipitant, also known as GW597599, is one of the most potent and selective NK(1) receptor antagonists ever discovered, showing appropriate pharmacokinetic properties and in vivo activity. Its actions support the utility of NK(1) receptor blockade in the alleviation of anxiety and, possibly, depression. It is under development as a potential antiemetic and anxiolytic drug, and as a treatment for tinnitusand insomnia.

化合物

SB 218795
Cat.No: T23316
Synonym:
Target: Neurokinin receptor
Senktide
Cat.No: T7633
Synonym:
Target: Neurokinin receptor
SB-222200
Cat.No: T16849
Synonym:
Target: Neurokinin receptor
Substance P
Cat.No: TP1087
Synonym: Neurokinin P,P物质
Target: Endogenous Metabolite, Neurokinin receptor
GR-73632
Cat.No: TP1572
Synonym:
Target: Neurokinin receptor
Maropitant
Cat.No: T7209
Synonym: 马罗匹坦,马罗皮坦
Target: Neurokinin receptor
Elinzanetant
Cat.No: T38144
Synonym:
Target: Neurokinin receptor
Fezolinetant
Cat.No: T15278
Synonym: ESN-364
Target: Neurokinin receptor
Talnetant
Cat.No: T7549
Synonym: SB 223412
Target: Neurokinin receptor
[Lys5,MeLeu9,Nle10]-NKA(4-10)
Cat.No: TP1883
Synonym:
Target: Neurokinin receptor
L-732138
Cat.No: T8235
Synonym:
Target: Neurokinin receptor
Tradipitant
Cat.No: T17156
Synonym: VLY-686,LY686017
Target: Neurokinin receptor
Substance P (7-11)
Cat.No: T7554
Synonym: Substance P 7-11(TFA)
Target: Others, Neurokinin receptor
Neurokinin A
Cat.No: TP1008
Synonym: α-Neurokinin,Substance K,神经激肽A,Neuromedin L
Target: Neurokinin receptor
Rolapitant
Cat.No: T3716
Synonym: 罗拉吡坦,SCH619734,罗拉匹坦
Target: Neurokinin receptor
Netupitant
Cat.No: T6905
Synonym: Ro 67-31898/000,奈妥吡坦,CID 6451149
Target: Neurokinin receptor
Vapreotide acetate
Cat.No: T13306L
Synonym: RC-160 acetate,醋酸伐普肽,BMY-41606 acetate
Target: Neurokinin receptor
Eprazinone dihydrochloride
Cat.No: T3034
Synonym: Resplen,Mucitux,Eftapan,NSC 317935,盐酸依普拉酮,依普拉酮二盐酸,Eprazinone 2HCl
Target: Others, Neurokinin receptor
Fosaprepitant dimeglumine
Cat.No: T1790
Synonym: 福沙匹坦二甲葡胺,L785298,福沙吡坦二甲葡胺,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
Aprepitant
Cat.No: T1743
Synonym: MK-869,MK-0869,阿瑞匹坦,L-754030,Aprepitant`
Target: HIV Protease, Antibacterial, Antibiotic, Neurokinin receptor
NK1 receptor antagonist 2
Cat.No: T72224
Synonym:
Target:
[Sar9,Met(O2)11]-Substance P
Cat.No: T7828
Synonym: Bhsar-sp,NA,精氨酰-脯氨酰-赖氨酰-脯氨酰-谷氨酰-谷氨酰-苯丙氨酰-苯丙氨酰-SAR-亮氨酸-蛋氨酸[O2]-胺
Target: Neurokinin receptor
Substance P(1-7)
Cat.No: T7396
Synonym: Substance P 1-7
Target: Others, Neurokinin receptor
Eledoisin Related Peptide
Cat.No: T7631
Synonym: Eledoisin RP,Eledoisin-Related Peptide,Eledoisin Related Peptide(2TFA)
Target: Neurokinin receptor
Neurokinin A(4-10)
Cat.No: T7559
Synonym: 神经激肽 A (4-10),Neurokinin A(4-10)(TFA)
Target: Neurokinin receptor
MEN 10207 acetate
Cat.No: T24446L
Synonym:
Target: Neurokinin receptor
Men 10376 TFA(135306-85-3,free)
Cat.No: TP1086
Synonym: Men 10376 TFA,Neurokinin-2 receptor antagonist TFA
Target: Neurokinin receptor
R 396 acetate
Cat.No: T24697L
Synonym:
Target: Neurokinin receptor
MEN11467
Cat.No: T12000
Synonym:
Target: Neurokinin receptor
Burapitant
Cat.No: T69140
Synonym: SSR 240600
Target: Neurokinin receptor
gamma-preprotachykinin amide (72-92) acetate
Cat.No: T9417L
Synonym: gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)
Target: Others
[Sar9] Substance P acetate(77128-75-7 free base)
Cat.No: TP1862L
Synonym:
Target: Neurokinin receptor
Men 10376
Cat.No: T16038
Synonym: Neurokinin-2 receptor antagonist
Target: CDK
[D-Trp2,7,9] Substance P
Cat.No: T76405
Synonym:
Target:
MEN-10612
Cat.No: T70496
Synonym:
Target:
TAC 363
Cat.No: T70243
Synonym:
Target:
NK-1 Antagonist 1
Cat.No: T12233
Synonym: Rolapitant intermediate
Target: Others
SCH 206272
Cat.No: T28706
Synonym: SCH206272,SCH-206272
Target:
GR 94800 TFA
Cat.No: T75880
Synonym:
Target:
MEN-10573
Cat.No: T70497
Synonym:
Target:
MDL-105212A HCl
Cat.No: T70295
Synonym:
Target:
YM44781
Cat.No: T29185
Synonym: YM 44781,YM-44781
Target:
Men 10376 TFA
Cat.No: T75879
Synonym:
Target:
YM49598
Cat.No: T29186
Synonym: YM-49598,YM 49598
Target:
NKP608
Cat.No: TQ0087
Synonym:
Target: Neurokinin receptor
Orvepitant maleate
Cat.No: T16406
Synonym: GW823296 maleate
Target: Neurokinin receptor
MEN-10354
Cat.No: T70689
Synonym:
Target:
GR 83074
Cat.No: T76431
Synonym:
Target:
Substance P (5-11)
Cat.No: T76454
Synonym:
Target:
Vestipitant
Cat.No: T69420
Synonym:
Target:
共73条,每页50条 1 2
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼